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Lead in PDB 6uwa: Mouse Pkc C1B and C2 Domains

Enzymatic activity of Mouse Pkc C1B and C2 Domains

All present enzymatic activity of Mouse Pkc C1B and C2 Domains:
2.7.11.13;

Protein crystallography data

The structure of Mouse Pkc C1B and C2 Domains, PDB code: 6uwa was solved by A.Aggarwal, J.Mire, J.C.Sacchettini, T.Igumenova, with X-Ray Crystallography technique. A brief refinement statistics is given in the table below:

Resolution Low / High (Å) 28.39 / 1.20
Space group P 21 21 21
Cell size a, b, c (Å), α, β, γ (°) 34.041, 58.974, 104.954, 90.00, 90.00, 90.00
R / Rfree (%) 13.4 / 15.3

Other elements in 6uwa:

The structure of Mouse Pkc C1B and C2 Domains also contains other interesting chemical elements:

Zinc (Zn) 2 atoms

Lead Binding Sites:

The binding sites of Lead atom in the Mouse Pkc C1B and C2 Domains (pdb code 6uwa). This binding sites where shown within 5.0 Angstroms radius around Lead atom.
In total 4 binding sites of Lead where determined in the Mouse Pkc C1B and C2 Domains, PDB code: 6uwa:
Jump to Lead binding site number: 1; 2; 3; 4;

Lead binding site 1 out of 4 in 6uwa

Go back to Lead Binding Sites List in 6uwa
Lead binding site 1 out of 4 in the Mouse Pkc C1B and C2 Domains


Mono view


Stereo pair view

A full contact list of Lead with other atoms in the Pb binding site number 1 of Mouse Pkc C1B and C2 Domains within 5.0Å range:
probe atom residue distance (Å) B Occ
A:Pb301

b:7.6
occ:0.95
OD1 A:ASP246 2.5 8.2 1.0
OD2 A:ASP187 2.5 9.0 1.0
OD2 A:ASP193 2.5 10.4 1.0
O A:TRP247 2.7 7.4 1.0
OD1 A:ASP187 2.7 9.0 1.0
OD1 A:ASP248 2.8 9.6 1.0
OD2 A:ASP246 2.8 8.6 1.0
CG A:ASP187 3.0 7.9 1.0
CG A:ASP246 3.0 7.2 1.0
CG A:ASP193 3.6 8.0 1.0
C A:TRP247 3.7 6.7 1.0
CG A:ASP248 3.8 8.5 1.0
CB A:ASP193 4.0 7.2 1.0
O A:HOH406 4.0 15.1 1.0
PB A:PB302 4.0 7.7 0.9
N A:ASP193 4.2 6.5 1.0
CA A:ASP248 4.2 7.4 1.0
N A:ASP248 4.3 7.1 1.0
O A:HOH484 4.4 15.7 1.0
CB A:ASP187 4.4 8.3 1.0
CB A:ASP246 4.5 7.0 1.0
OD2 A:ASP248 4.5 8.3 1.0
N A:TRP247 4.6 6.4 1.0
CB A:ASP248 4.6 6.8 1.0
OD1 A:ASP193 4.6 9.7 1.0
C A:ASP246 4.7 6.2 1.0
CA A:ASP193 4.7 6.4 1.0
C A:SER192 4.8 6.7 1.0
CA A:TRP247 4.8 6.8 1.0
CA A:SER192 4.8 6.6 1.0
O A:HOH499 4.9 26.6 1.0
O A:ASP246 5.0 7.2 1.0
O4 A:CIT308 5.0 14.5 1.0

Lead binding site 2 out of 4 in 6uwa

Go back to Lead Binding Sites List in 6uwa
Lead binding site 2 out of 4 in the Mouse Pkc C1B and C2 Domains


Mono view


Stereo pair view

A full contact list of Lead with other atoms in the Pb binding site number 2 of Mouse Pkc C1B and C2 Domains within 5.0Å range:
probe atom residue distance (Å) B Occ
A:Pb302

b:7.7
occ:0.93
O6 A:CIT308 2.5 11.7 1.0
OD1 A:ASP248 2.5 9.6 1.0
OD2 A:ASP248 2.6 8.3 1.0
OD1 A:ASP187 2.6 9.0 1.0
O7 A:CIT308 2.7 11.4 1.0
OD2 A:ASP254 2.8 8.6 1.0
O2 A:CIT308 2.8 12.1 1.0
OD2 A:ASP246 2.8 8.6 1.0
O A:MET186 2.8 8.6 1.0
CG A:ASP248 2.9 8.5 1.0
C6 A:CIT308 3.4 10.8 1.0
C1 A:CIT308 3.5 11.7 1.0
C3 A:CIT308 3.5 11.5 1.0
C A:MET186 3.7 7.3 1.0
CG A:ASP254 3.7 7.0 1.0
CG A:ASP187 3.8 7.9 1.0
PB A:PB301 4.0 7.6 0.9
PB A:PB304 4.1 7.5 0.9
CG A:ASP246 4.1 7.2 1.0
CB A:MET186 4.1 7.5 1.0
C2 A:CIT308 4.1 11.2 1.0
PB A:PB303 4.3 8.3 0.9
O1 A:CIT308 4.3 11.1 1.0
CA A:ASP187 4.3 8.2 1.0
N A:ASP187 4.3 7.3 1.0
OD1 A:ASP254 4.3 7.8 1.0
CB A:ASP248 4.4 6.8 1.0
O4 A:CIT308 4.4 14.5 1.0
O A:HOH406 4.5 15.1 1.0
O5 A:CIT308 4.5 13.2 1.0
OD2 A:ASP187 4.5 9.0 1.0
CB A:ASP254 4.5 7.0 1.0
CA A:MET186 4.6 7.9 1.0
CB A:ASP187 4.6 8.3 1.0
OD1 A:ASP246 4.8 8.2 1.0
C4 A:CIT308 4.9 13.4 1.0

Lead binding site 3 out of 4 in 6uwa

Go back to Lead Binding Sites List in 6uwa
Lead binding site 3 out of 4 in the Mouse Pkc C1B and C2 Domains


Mono view


Stereo pair view

A full contact list of Lead with other atoms in the Pb binding site number 3 of Mouse Pkc C1B and C2 Domains within 5.0Å range:
probe atom residue distance (Å) B Occ
A:Pb303

b:8.3
occ:0.91
O2 A:CIT308 2.4 12.1 1.0
O2 A:CIT309 2.5 8.6 1.0
O1 A:CIT309 2.6 9.1 1.0
OD2 A:ASP254 2.6 8.6 1.0
O1 A:CIT308 2.6 11.1 1.0
C1 A:CIT308 2.9 11.7 1.0
C1 A:CIT309 2.9 8.5 1.0
SG A:CYS143 3.4 7.4 1.0
SG A:CYS118 3.4 7.8 1.0
CG A:ASP254 3.4 7.0 1.0
CB A:CYS118 3.7 8.4 1.0
O A:MET186 3.9 8.6 1.0
OD1 A:ASP254 3.9 7.8 1.0
ZN A:ZN310 3.9 7.0 1.0
O A:HOH539 4.1 9.9 1.0
PB A:PB304 4.2 7.5 0.9
PB A:PB302 4.3 7.7 0.9
C2 A:CIT308 4.4 11.2 1.0
C2 A:CIT309 4.4 7.8 1.0
CB A:ASP254 4.5 7.0 1.0
ND1 A:HIS140 4.7 7.3 1.0
CG A:GLN142 4.8 9.1 1.0
SD A:MET186 4.9 10.4 1.0
C A:MET186 5.0 7.3 1.0
O A:HOH469 5.0 13.6 1.0

Lead binding site 4 out of 4 in 6uwa

Go back to Lead Binding Sites List in 6uwa
Lead binding site 4 out of 4 in the Mouse Pkc C1B and C2 Domains


Mono view


Stereo pair view

A full contact list of Lead with other atoms in the Pb binding site number 4 of Mouse Pkc C1B and C2 Domains within 5.0Å range:
probe atom residue distance (Å) B Occ
A:Pb304

b:7.5
occ:0.94
OD1 A:ASP254 2.4 7.8 1.0
O6 A:CIT309 2.4 8.0 1.0
O A:ARG252 2.5 8.0 1.0
O2 A:CIT309 2.7 8.6 1.0
O7 A:CIT309 2.7 8.0 1.0
OD2 A:ASP248 2.8 8.3 1.0
OG1 A:THR251 3.1 10.1 1.0
CG A:ASP254 3.1 7.0 1.0
C6 A:CIT309 3.2 7.4 1.0
OD2 A:ASP254 3.3 8.6 1.0
O6 A:CIT308 3.3 11.7 1.0
O2 A:CIT308 3.3 12.1 1.0
C3 A:CIT309 3.5 7.8 1.0
C1 A:CIT309 3.6 8.5 1.0
C A:ARG252 3.6 7.0 1.0
CG A:ASP248 3.7 8.5 1.0
C6 A:CIT308 3.9 10.8 1.0
CB A:THR251 4.0 9.6 1.0
O5 A:CIT308 4.0 13.2 1.0
PB A:PB302 4.1 7.7 0.9
N A:ARG252 4.1 7.3 1.0
C2 A:CIT309 4.1 7.8 1.0
CB A:ASP248 4.2 6.8 1.0
PB A:PB303 4.2 8.3 0.9
O4 A:CIT309 4.4 11.1 1.0
O5 A:CIT309 4.4 7.8 1.0
CA A:ARG252 4.4 6.8 1.0
C A:THR251 4.4 7.6 1.0
C1 A:CIT308 4.5 11.7 1.0
O A:HOH460 4.5 9.1 1.0
O1 A:CIT309 4.6 9.1 1.0
CB A:ASP254 4.6 7.0 1.0
OD1 A:ASP248 4.6 9.6 1.0
C A:ASN253 4.7 6.4 1.0
N A:ASN253 4.7 6.8 1.0
N A:ASP254 4.7 6.1 1.0
O A:HOH532 4.7 23.0 1.0
CB A:ARG252 4.8 7.7 1.0
CA A:ASN253 4.8 7.3 1.0
C4 A:CIT309 4.8 8.4 1.0
CA A:THR251 4.8 8.5 1.0
O A:THR251 4.9 8.4 1.0
O A:ASN253 4.9 6.6 1.0

Reference:

T.Igumenova, A.Aggarwal, J.Mire, J.C.Sacchettini, T.Igumenova. N/A N/A.
Page generated: Wed Dec 16 02:02:30 2020

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